• Fluorophore labeled kinase detects ligands that bind within the MAPK insert of p38α kinase 

      Getlik, Matthaus; Simard, Jeffrey R.; Termathe, Martin; Grutter, Christian; Rabiller, Matthias; Van Otterlo, Willem A. L.; Rauh, Daniel (Public Library of Science, 2012-07-02)
      ENGLISH ABSTRACT: The vast majority of small molecules known to modulate kinase activity, target the highly conserved ATP-pocket. Consequently, such ligands are often less specific and in case of inhibitors, this leads to ...